XALKORI

GrowthSM

crizotinib

NDAORALCAPSULE, PELLETS
Approved
Sep 2023
Lifecycle
Growth
Competitive Pressure
8/100
Clinical Trials
20

Mechanism of Action

Cytochrome P450 3A Inhibitors

Pharmacologic Class:

Kinase Inhibitor

Clinical Trials (5)

NCT06140836Phase 3Active Not Recruiting

A Study of Repotrectinib Versus Crizotinib in Participants With Locally Advanced or Metastatic Tyrosine Kinase Inhibitor (TKI)-naïve ROS1-positive Non-Small Cell Lung Cancer (NSCLC) (TRIDENT-3)

Started Dec 2023
190 enrolled
Carcinoma, Non-Small-Cell Lung
NCT05987332Phase 2/3Active Not Recruiting

IDE196 (Darovasertib) in Combination With Crizotinib as First-line Therapy in Metastatic Uveal Melanoma

Started Oct 2023
420 enrolled
Metastatic Uveal Melanoma
NCT06569420Phase 3Active Not Recruiting

Study Of Comparing SAF-189s With Crizotinib In First Line ALK-Positive Advanced and Metastatic NSCLC

Started Dec 2021
275 enrolled
Non-Small Cell Lung CancerALK-positiveSAF-189s
NCT04603807Phase 3Active Not Recruiting

A Study to Compare the Efficacy and Safety of Entrectinib and Crizotinib in Participants With Advanced or Metastatic ROS1 Non-small Cell Lung Cancer (NSCLC) With and Without Central Nervous System (CNS) Metastases

Started Sep 2021
220 enrolled
Carcinoma, Non-Small-Cell Lung
NCT04856293Phase 1Completed

Bioequivalence Study for Crizotinib Encapsulated Microsphere Formulation (eMS)

Started Apr 2021
25 enrolled
Healthy Participants

Loss of Exclusivity

LOE Date
Nov 6, 2029
44 months away
Patent Expiry
Nov 6, 2029

Patent Records (3)

Patent #ExpiryTypeUse Code
7825137
May 12, 2027
U-3058
7858643
Oct 8, 2029
SubstanceProduct
8217057
Nov 6, 2029
Substance