KOSELUGO

PeakSM

selumetinib

NDAORALCAPSULEPriority Review
Approved
Apr 2020
Lifecycle
Peak
Competitive Pressure
8/100
Clinical Trials
20

Mechanism of Action

Mitogen-Activated Protein Kinase Kinase 1 Inhibitors

Pharmacologic Class:

Kinase Inhibitor

Clinical Trials (5)

NCT06502171Phase 1Not Yet Recruiting

Study of Cabozantinib With Selumetinib for Plexiform Neurofibromas

Started Aug 2026
30 enrolled
Neurofibromatosis 1Plexiform Neurofibroma
NCT06360406N/ARecruiting

Real-World Treatment Study of Koselugo (Selumetinib)

Started Jun 2024
200 enrolled
Neurofibromatosis 1Neurofibroma, Plexiform
NCT06175637N/AActive Not Recruiting

Observational Study to Evaluate the Effect and Safety of Selumetinib in Pediatric Patients With NF1-PNs

Started Dec 2023
409 enrolled
Neurofibroma, Plexiform
NCT05825365Phase 2Withdrawn

Selumetinib in Chinese Paediatric With Post-operative NF1-PNs, PhaseⅡ, Double-Blinded, Placebo-Controlled Study

Started Aug 2023
0
Neurofibromatosis Type 1Plexiform NeurofibromasPost-operative
NCT05891847N/AActive Not Recruiting

Non-interventional Study of Patients With PN NF1 Starting Selumetinib in Russia

Started Mar 2023
150 enrolled
Neurofibroma

Loss of Exclusivity

LOE Date
Mar 26, 2029
37 months away
Patent Expiry
Mar 26, 2029
Exclusivity Expiry
Nov 19, 2028

Patent Records (5)

Patent #ExpiryTypeUse Code
8178693
Mar 13, 2026
SubstanceProduct
9562017
Dec 12, 2026
Substance
U-4357
9156795
Dec 12, 2026
SubstanceProduct
7425637
Mar 13, 2028
Substance
11813246
Mar 26, 2029
Product