GAVRETO

PeakSM

pralsetinib

NDAORALCAPSULEPriority Review
Approved
Sep 2020
Lifecycle
Peak
Competitive Pressure
0/100
Clinical Trials
5

Mechanism of Action

Rearranged during Transfection (RET) Inhibitors

Pharmacologic Class:

Kinase Inhibitor

Clinical Trials (5)

NCT04760288Phase 3Withdrawn

A Study of Pralsetinib Versus Standard of Care (SOC) for Treatment of RET-Mutated Medullary Thyroid Cancer (MTC).

Started Nov 2023
0
Medullary Thyroid Cancer
NCT04697446N/AUnknown

External Control, Observational, Retrospective Study Comparing Pralsetinib to Best Available Therapy in Patients With RET-Fusion Positive NSCLC

Started Dec 2020
279 enrolled
RET-fusion Non Small Cell Lung CancerLung NeoplasmCarcinoma, Non-Small-Cell Lung+14 more
NCT04222972Phase 3Terminated

A Study of Pralsetinib Versus Standard of Care for First-Line Treatment of Advanced Non-Small Cell Lung Cancer (NSCLC)

Started Jul 2020
223 enrolled
RET-fusion Non Small Cell Lung CancerLung NeoplasmCarcinoma, Non-Small-Cell Lung+14 more
NCT03037385Phase 1/2Completed

Phase 1/2 Study of the Highly-selective RET Inhibitor, Pralsetinib (BLU-667), in Participants With Thyroid Cancer, Non-Small Cell Lung Cancer, and Other Advanced Solid Tumors

Started Mar 2017
590 enrolled
RET-altered Non Small Cell Lung CancerMedullary Thyroid CancerRET-altered Papillary Thyroid Cancer+37 more
NCT04204928N/AApproved For Marketing

Pre-Approval Access Program (PAAP) for Pralsetinib (BLU-667) in Patients With Unresectable or Metastatic NSCLC or MTC

Non-Small Cell Lung CancerMedullary Thyroid Cancer

Loss of Exclusivity

LOE Date
Jul 7, 2042
199 months away
Patent Expiry
Jul 7, 2042
Exclusivity Expiry
Dec 1, 2027

Patent Records (5)

Patent #ExpiryTypeUse Code
10030005
Nov 1, 2036
SubstanceProduct
U-3002
11273160
Apr 3, 2039
U-2952
11872192
Apr 3, 2039
U-2952
11963958
Apr 3, 2039
U-2828
12539303
Apr 3, 2039
U-2828