ZORYVE

Peak

roflumilast

NDATOPICALCREAM
Approved
Jul 2022
Lifecycle
Peak
Competitive Pressure
0/100
Clinical Trials
20

Mechanism of Action

Phosphodiesterase 4 Inhibitors

Pharmacologic Class:

Phosphodiesterase 4 Inhibitor

Clinical Trials (5)

NCT02671942Phase 2Terminated

A Multicenter Randomized Double-blind Clinical Study Evaluated the Safety, Pharmacokinetic and Pharmacodynamic Characteristics of Roflumilast in COPD Patients

Started Mar 2016
NCT02165826Phase 3Completed

Evaluation of Tolerability and Pharmacokinetics of Roflumilast, 250μg and 500μg, as add-on to Standard COPD Treatment to Treat Severe COPD

Started May 2014
1,323 enrolled
Chronic Obstructive Pulmonary Disease (COPD)
NCT02079844Phase 1Completed

Roflumilast Plus Antipsychotics Proof of Mechanism Study in Schizophrenia

Started Mar 2014
20 enrolled
Schizophrenia
NCT02051335Phase 1Completed

Roflumilast and Donepezil to Reverse Scopolamine Induced Cognitive Deficits in Healthy Adults

Started Jan 2014
27 enrolled
Memory ImpairmentAlzheimer's Disease
NCT03381573N/ACompleted

Long-term Observational Study of the Safety of Roflumilast

Started Dec 2013
135,856 enrolled
COPD

Loss of Exclusivity

LOE Date
Aug 25, 2037
139 months away
Patent Expiry
Aug 25, 2037
Exclusivity Expiry
Oct 4, 2028

Patent Records (5)

Patent #ExpiryTypeUse Code
9907788
Jun 7, 2037
U-3970
10940142
Jun 7, 2037
Product
11793796
Jun 7, 2037
Product
11819496
Jun 7, 2037
U-3748
11992480
Jun 7, 2037
U-3748