XTANDI

Peak

enzalutamide

NDAORALCAPSULEPriority Review
Approved
Aug 2012
Lifecycle
Peak
Competitive Pressure
0/100
Clinical Trials
20

Mechanism of Action

Androgen Receptor Antagonists

Pharmacologic Class:

Androgen Receptor Inhibitor

Clinical Trials (5)

NCT06616155Phase 1/2Recruiting

Ruxolitinib and Enzalutamide for the Treatment of Metastatic Castration-Resistant Prostate Cancer

Started Jan 2026
39 enrolled
Castration-Resistant Prostate CarcinomaMetastatic Prostate AdenocarcinomaStage IVB Prostate Cancer AJCC v8
NCT06844383Phase 2Recruiting

A Study of Talazoparib With or Without Enzalutamide in People With Prostate Cancer Who Have Previously Received Abiraterone Acetate

Started Oct 2025
126 enrolled
Prostate Cancer (Adenocarcinoma)mCRPC (Metastatic Castration-resistant Prostate Cancer)
NCT07028853Phase 3Recruiting

This Study Will Explore Whether a Combination of the Investigational Drug Mevrometostat (PF-06821497) and Enzalutamide Will Work Better Than Taking Enzalutamide Alone in Participants With mCSPC Who Are ARPI naïve.

Started Sep 2025
1,000 enrolled
Metastatic Castration Sensitive Prostate Cancer (mCSPC)Hormone Sensitive Prostate CancerProstate Cancer+1 more
NCT07086651N/ACompleted

A Study to Learn About Two Medicines (Apalutamide and Enzalutamide) in People With Metastatic Castration-sensitive Prostate Cancer (mCSPC)

Started Jul 2025
1,300 enrolled
Metastatic Castration Sensitive Prostate Cancer (mCSPC)Cancer of the ProstateProstate Neoplasms+1 more
NCT06130995Phase 1Recruiting

Relugolix + Enzalutamide Study in High-Risk Prostate Cancer

Started Dec 2024
46 enrolled
Androgen Deprivation TherapyLocally Advanced Prostate Cancer

Loss of Exclusivity

LOE Date
Feb 23, 2037
133 months away
Patent Expiry
Feb 23, 2037
Exclusivity Expiry
Nov 17, 2026

Patent Records (4)

Patent #ExpiryTypeUse Code
9126941
May 15, 2026
U-3763
8183274
Aug 24, 2026
U-3763
7709517
Aug 13, 2027
SubstanceProduct
12161628
Feb 23, 2037
U-4104