VANRAFIA

Launch

atrasentan

NDAORALTABLET
Approved
Apr 2025
Lifecycle
Launch
Competitive Pressure
0/100
Clinical Trials
15

Mechanism of Action

(Ki = 0.034 nM) with >1800-fold selectivity for the ET A receptor compared to the endothelin type B receptor (Ki = 63.3 nM). Endothelin (ET)-1 is thought to contribute to the pathogenesis of IgAN via the ET A R.

Clinical Trials (5)

NCT05834738Phase 2Completed

Randomized, Double-blind, Placebo-controlled, Crossover Study of Atrasentan in Subjects With IgA Nephropathy

Started Jul 2023
54 enrolled
IgA NephropathyImmunoglobulin A Nephropathy
NCT04573920Phase 2Active Not Recruiting

Atrasentan in Patients With Proteinuric Glomerular Diseases

Started Mar 2021
103 enrolled
IgA NephropathyFocal Segmental GlomerulosclerosisAlport Syndrome+3 more
NCT02118714Phase 2Completed

Atrasentan Spermatogenesis and Testicular Function

Started Apr 2015
20 enrolled
NephropathyDiabetes
NCT01858532Phase 3Terminated

Study Of Diabetic Nephropathy With Atrasentan

Started May 2013
5,107 enrolled
Diabetic Nephropathy
NCT01424319Phase 2Completed

Reducing Residual Albuminuria in Subjects With Diabetes and Nephropathy With Atrasentan

Started Aug 2011
58 enrolled
Chronic Kidney DiseaseDiabetic Nephropathy

Loss of Exclusivity

LOE Date
Feb 23, 2041
182 months away
Patent Expiry
Feb 23, 2041
Exclusivity Expiry
Apr 2, 2030

Patent Records (5)

Patent #ExpiryTypeUse Code
8623819
Aug 22, 2028
U-3980
11874283
Feb 18, 2032
U-3980
10016393
Jul 7, 2034
Product
9364458
Jul 7, 2034
Product
U-3980
12121509
Dec 16, 2040
U-3980