TURALIO

Peak

pexidartinib hydrochloride

NDAORALCAPSULEPriority Review
Approved
Aug 2019
Lifecycle
Peak
Competitive Pressure
0/100
Clinical Trials
3

Mechanism of Action

1 receptor (CSF1R), KIT proto-oncogene receptor tyrosine kinase (KIT), and FMS-like tyrosine kinase 3 (FLT3) harboring an internal tandem duplication (ITD) mutation. Overexpression of the CSF1R ligand promotes cell proliferation and accumulation in the synovium. In vitro, pexidartinib inhibited…

Clinical Trials (3)

NCT04635111N/ARecruiting

A Long-term Study Evaluating Hepatotoxicity Associated With TURALIO™ (Pexidartinib) Treatment

Started Jan 2021
30 enrolled
HepatotoxicityTenosynovial Giant Cell Tumor
NCT04526704Phase 4Completed

Study to Evaluate Discontinuation and Re-Treatment in Participants With Tenosynovial Giant Cell Tumor (TGCT) Previously Treated With Pexidartinib

Started Oct 2020
32 enrolled
Tenosynovial Giant Cell Tumor
NCT04488822Phase 3Active Not Recruiting

A Study of the Efficacy and Safety of Pexidartinib in Adult Subjects With TGCT

Started Sep 2020
40 enrolled
Tenosynovial Giant Cell Tumor

Loss of Exclusivity

LOE Date
Jul 24, 2038
150 months away
Patent Expiry
Jul 24, 2038
Exclusivity Expiry
Aug 2, 2026

Patent Records (5)

Patent #ExpiryTypeUse Code
8404700
Nov 21, 2027
Substance
9169250
Nov 21, 2027
Substance
8722702
Nov 21, 2027
Substance
8461169
Apr 19, 2028
U-2606
7893075
May 4, 2033
Substance