ORLADEYO

Peak

berotralstat hydrochloride

NDAORALCAPSULE
Approved
Dec 2020
Lifecycle
Peak
Competitive Pressure
0/100

Mechanism of Action

activity. Plasma kallikrein is a protease that cleaves high-molecular-weight kininogen (HMWK) to generate cleaved HMWK (cHMWK) and bradykinin, a potent vasodilator that increases vascular permeability resulting in swelling and pain associated with HAE. In patients with HAE due to C1-inhibitor…

Loss of Exclusivity

LOE Date
May 1, 2040
172 months away
Patent Expiry
May 1, 2040
Exclusivity Expiry
Jun 3, 2028

Patent Records (5)

Patent #ExpiryTypeUse Code
10689346
Mar 9, 2035
U-3010
11708333
Mar 9, 2035
U-3300
10329260
Mar 9, 2035
Substance
12116346
Mar 9, 2035
Substance
11230530
Mar 9, 2035
U-3300