GALLIUM GA 68 EDOTREOTIDE

PeakPeptide

edotreotide gallium ga-68

NDAINTRAVENOUSSOLUTION
Approved
Aug 2019
Lifecycle
Peak
Competitive Pressure
30/100

Mechanism of Action

68 DOTATOC binds to somatostatin receptors, with highest affinity (K i = 2.5± 0.5 nanomolar) for subtype 2 receptors (sstr2). Ga 68 DOTATOC binds to cells that express somatostatin receptors including malignant neuroendocrine cells, which overexpress sstr2 receptors. Gallium 68 is a β+ emitting…