FANAPT

Peak

iloperidone

NDAORALTABLET
Approved
May 2009
Lifecycle
Peak
Competitive Pressure
0/100
Clinical Trials
19

Mechanism of Action

unknown. However, the efficacy of iloperidone could be mediated through a combination of dopamine type 2 (D 2 ) and serotonin type 2 (5-HT 2 ) antagonism. Iloperidone forms an active metabolite, P88, that has an in vitro receptor binding profile similar to the parent drug.

Pharmacologic Class:

Atypical Antipsychotic

Indications (1)

Clinical Trials (5)

NCT07090161Phase 2Recruiting

Evaluation of Efficacy and Safety of Iloperidone for the Treatment of Participants With Uncontrolled Hypertension

Started Sep 2025
240 enrolled
HypertensionUncontrolled Hypertension
NCT06494397Phase 1Completed

Pharmacokinetic Study of VHX-896 and Iloperidone Tablets Under Steady-State Conditions

Started Jul 2024
26 enrolled
SchizophreniaBipolar I Disorder
NCT05648591Phase 4Recruiting

Safety and Tolerability of Open-Labeled Iloperidone in Adolescents

Started May 2023
100 enrolled
SchizophreniaBipolar I Disorder
NCT05344365Phase 2Withdrawn

A Study to Evaluate Iloperidone for the Treatment of Parkinson's Disease Psychosis

Started Jun 2022
0
Parkinson Disease Psychosis
NCT04969211Phase 1Completed

Bioequivalence Study Between VHX-896 Tablets and Iloperidone Tablets in Healthy Volunteers

Started Jun 2021
25 enrolled
Healthy

Loss of Exclusivity

LOE Date
Dec 28, 2031
70 months away
Patent Expiry
Dec 28, 2031
Exclusivity Expiry
Apr 2, 2027

Patent Records (5)

Patent #ExpiryTypeUse Code
8586610
Nov 2, 2027
U-1625
9157121
Apr 5, 2030
U-1674
8652776
Aug 31, 2030
U-1685
8999638
Oct 28, 2030
U-1674
9074255
Dec 17, 2030
U-1674