AYVAKIT

PeakSM

avapritinib

NDAORALTABLETPriority Review
Approved
Jan 2020
Lifecycle
Peak
Competitive Pressure
0/100
Clinical Trials
11

Mechanism of Action

Tyrosine Kinase Inhibitors

Pharmacologic Class:

Kinase Inhibitor

Clinical Trials (5)

NCT06748001Phase 4Recruiting

Avapritinib Rollover Study

Started Nov 2024
60 enrolled
Mastocytosis, Systemic
NCT06327685Phase 1Recruiting

Avapritinib With Decitabine in Patients With SM-AHN

Started Mar 2024
34 enrolled
Systemic Mastocytosis With an Associated Hematologic Neoplasm
NCT04908176Phase 1Completed

A Drug-drug Interaction Study of Avapritinib and Midazolam

Started Aug 2022
10 enrolled
Gastrointestinal Stromal TumorsGISTNon-resectable Advanced Solid Tumors+1 more
NCT04773782Phase 1/2Completed

A Study of Avapritinib in Pediatric Patients With Solid Tumors Dependent on KIT or PDGFRA Signaling

Started Feb 2022
29 enrolled
Solid Tumor, Unspecified, ChildRelapsed Solid NeoplasmCNS Tumor
NCT04825574Phase 4Completed

Study for Patients Previously Treated in Avapritinib Clinical Trials

Started May 2021
2 enrolled
Gastrointestinal Stromal Tumors

Loss of Exclusivity

LOE Date
Mar 8, 2042
194 months away
Patent Expiry
Mar 8, 2042
Exclusivity Expiry
May 22, 2030

Patent Records (5)

Patent #ExpiryTypeUse Code
11827642
Oct 15, 2034
SubstanceProduct
U-3506
9200002
Oct 15, 2034
SubstanceProduct
U-3506
9944651
Oct 15, 2034
SubstanceProduct
U-3506
9994575
Oct 15, 2034
SubstanceProduct
U-3506
12252494
Apr 10, 2040
U-3506