APREMILAST

Post-LOE

apremilast

ANDAORALTABLET
Approved
Apr 2023
Lifecycle
Post-LOE
Competitive Pressure
30/100
Clinical Trials
20

Mechanism of Action

4 (PDE4) specific for cyclic adenosine monophosphate (cAMP). PDE4 inhibition results in increased intracellular cAMP levels. The specific mechanism(s) by which apremilast exerts its therapeutic action is not well defined.

Clinical Trials (5)

NCT06122649Phase 3Completed

A Study to Investigate Efficacy and Safety of Apremilast 30 mg Twice Daily (BID) in Chinese Participants With Moderate to Severe Plaque-type Psoriasis (PsO)

Started Nov 2023
203 enrolled
Plaque Psoriasis
NCT06088199Phase 3Active Not Recruiting

A Study of Apremilast in Pediatric Participants in Children With Mild to Moderate Plaque Psoriasis

Started Oct 2023
51 enrolled
Plaque Psoriasis
NCT05767047Phase 3Recruiting

A Study of Apremilast in Children With Oral Ulcers Associated With Behçet's Disease or Juvenile Psoriatic Arthritis

Started Mar 2023
48 enrolled
Behçet's DiseaseJuvenile Psoriatic Arthritis
NCT05565560Phase 3Active Not Recruiting

A Study to Assess the Efficacy and Safety of Apremilast in Japanese Pediatric Participants With Moderate to Severe Plaque Psoriasis

Started Jan 2023
17 enrolled
Plaque Psoriasis
NCT05744466N/ARecruiting

A Real-world Observational Study to Compare Effectiveness of Deucravacitinib Vs Apremilast in Adults With Plaque Psoriasis

Started Sep 2022
1,500 enrolled
Psoriasis