ALVIMOPAN (alvimopan) by Pfizer is μ-opioid receptor with a ki of 0. First approved in 2023.
Drug data last refreshed 18h ago
μ-opioid receptor with a Ki of 0.4 nM (0.2 ng/mL) and no measurable opioid-agonist effects in standard pharmacologic assays. The dissociation of [H]-alvimopan from the human μ-opioid receptor is slower than that of other opioid ligands, consistent with its higher affinity for the receptor. At…
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Indication data is being enriched from DailyMed and FDA labeling. Check back soon for approved therapeutic uses.
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